Carbetocin acetate
Description
Carbetocin acetate, an oxytocin (OT) analogue, is an oxytocin receptor agonist with a Ki of 7.1 nM. Carbetocin acetate has high affinity to chimeric N-terminus (E1) of the oxytocin receptor (Ki=1.17 ??M). Carbetocin acetate has the potential for postpartum hemorrhage research. Carbetocin acetate can crosse the blood-brain barrier and produces antidepressant-like activity via activation of oxytocin receptors in the CNS.
Product Information
| Product Name | Carbetocin acetate |
| Molecular Weight | 1048.21 |
| Formula | C47H73N11O14S |
| CAS Number | 1631754-28-3 |
| Appearance | Solid |
| Color | White to off-white |
| Sequence | {Butyric acid}-Tyr(OMe)-Ile-Gln-Asn-Cys-Pro-Leu-Gly-NH2 (carba sulfide bridge:Butyric acid1-Cys6) |
| Sequence Shortening | {Butyric acid}-Tyr(OMe)-IIQNCPLG-NH2 (carba sulfide bridge:Butyric acid1-Cys6) |
| Storage | Sealed storage, away from moisture and light, under nitrogen Powder -80??C 2 years -20??C 1 year *In solvent : -80??C, 6 months; -20??C, 1 month (sealed storage, away from moisture and light, under nitrogen) |
